In this article, I’m going to teach you how to use phenibut for opiate withdrawal. Phenibut is a truly incredible natural supplement that has powerful relaxation, sleep-inducing, and mood-enhancing effects. I just learned about phenibut a few months ago, and after trying it out on myself a few times, I’ve put together an effective phenibut for opiate withdrawal protocol that is easy to follow and inexpensive.
If you’re interested in learning about phenibut for opiate withdrawal and how you can use it safely, you’ve come to the right place.
I’m going to cover the following key points:
- Phenibut history
- How phenibut works in the body
- My experience with phenibut
- How to use phenibut for opiate withdrawal
- Phenibut side effects and precautions
- Where to purchase phenibut
Table of Contents
A Brief History of Phenibut
Phenibut is a neuropsychotropic drug that was discovered in Russia in the 1960’s. In 1975 phenibut was incorporated into the Russian cosmonauts’ kit for individuals who participated in the Apollo-Soyuz joint mission. Since conventional tranquilizers for stress and anxiety can lead to feelings of drowsiness (not cool for people in spacecrafts), phenibut was mandated to be included in the Russian cosmonauts’ medical kit.
Note: Phenibut is widely used in Russia to relieve tension, anxiety, fear, to improve sleep, and as a pre- or post-operative medication. Phenibut is also used to treat depression and PTSD.
How Phenibut Works in the Body
Phenibut is a Central Nervous System (CNS) depressant and derivative of gamma-aminobutyric acid (GABA). GABA is an inhibitory neurotransmitter that produces feelings of calmness and tranquility. GABA inhibits nerve transmission in the brain, thus calming nervous activity.
I often refer to GABA as the brain’s “natural Valium”. However, since Valium and other anxiolytic (anti-anxiety) medications in the benzodiazepine class of drugs bind to GABA receptors, one could also refer to Valium as “unnatural GABA”.
GABA is sold in supplement form, though the general consensus is that GABA supplements cannot penetrate the Blood Brain Barrier (BBB), so their efficacy is questionable. However, the Russian chemists found a way to create GABA-like supplements that can cross the BBB and function like GABA in the brain.
Beta-phenyl-gamma-aminobutyric acid HCL, also known as phenibut, is a designer GABA analogue. Phenibut is the result of chemists adding a 6-carbon ring to the GABA supplement, thus allowing phenibut to effectively cross the barrier and act on GABA receptors.
Phenibut has anxiolytic and nootropic (cognition-enhancing) effects. Phenibut acts directly on the GABAB receptor sites. Drugs and substances such as baclofen, GHB, and alcohol also bind to these sites. Some believe that high doses of phenibut also bind to the GABAA receptors, which is where benzodiazepine drugs such as Valium, Ativan, Klonopin, and Xanax bind to, though this is a topic of debate in the scientific community.
Note: Another exciting aspect of phenibut is it’s stimulating action on dopamine receptors, which causes an increase of dopamine, a key neurotransmitter for feeling pleasure, happiness and motivation.
Phenibut supplementation can lead to the following benefits:
- Mental and physical relaxation
- Enhanced mood
- Sleep induction
- Reduction of stress
My Experience with Phenibut
When I first learned about phenibut for opiate withdrawal a few months ago, I decided to try some out on myself from a strictly investigative perspective. My goal was to try a few different dosages to see what could work best for opiate withdrawal anxiety and insomnia. I quit Rx opiates and heroin years ago, but even though I wasn’t using phenibut for opiate withdrawal, I feel like I found a great dosage that can work well for most individuals.
First I tried 500 mg of phenibut. Phenibut, unlike most supplements or drugs, comes on very slow. The typical duration for phenibut to achieve peak effects is four hours, and I felt my first dose around two hours in, with it peaking at about four hours. I felt a deep relaxation in my body and mind, and the tranquility stayed with me throughout the day, ending in a very restful sleep.
Note: The next time I used 1,000 mg of phenibut. It was way too strong for me! I felt this “out of synch with reality” feeling. Yes, I was relaxed, but I didn’t have the pleasant nootropic benefits I received from the 500 mg dose. However, this higher dose could be very beneficial for opiate withdrawal-induced anxiety. Also, due to biochemical uniqueness and GABA tolerance, optimal dosages will vary between individuals.
How to Use Phenibut for Opiate Withdrawal
Based on my in-depth research, as well as my personal use of the supplement, I’ve come up with some phenibut for opiate withdrawal dosing guidelines that you will benefit from adhering to.
Phenibut for opiate withdrawal dosing:
- Dosages of phenibut may vary depending on the individual’s GABA tolerance and sensitivity.
- Start with a low dosage of 250 mg to test your tolerance to phenibut.
- After 4 hours, if you don’t feel the effects take another 500 mg.
- During the day take between 250-500 mg of phenibut per dose for opiate withdrawal anxiety.
- A few hours before bedtime, take up to 500 mg of phenibut for opiate withdrawal insomnia.
- Only use phenibut for opiate withdrawal a maximum of 3 days, otherwise, you can experience phenibut withdrawal symptoms (you can avoid this by continually cycling phenibut 3 days on, 3 days off).
- Phenibut’s half-life is approx. 5-6 hours.
- Do not redose anytime before the 4-hour mark.
Note: Phenibut comes in crystals or powder. Some brands have them already in capsules, but they are more expensive. It’s cheaper to purchase it loose and either mix it with a beverage of your choice or put them in your own capsules to avoid the unpleasant taste.
Possible phenibut side effects include:
- Memory reduction
- Gastrointestinal (GI) distress
- Lowered inhibitions
- Mixing phenibut with other GABAergics is dangerous.
- Mixing phenibut with GHB, alcohol, and benzodiazepines can lead to respiratory depression and death.
- Phenibut should not be used by individuals with Parkinson’s disease.
Where to Purchase Phenibut for Opiate Withdrawal
Depending on what country you live in, phenibut may be considered a prescription-only drug, an over-the-counter drug, or a dietary supplement. Presently in the USA, phenibut is legally sold as a dietary supplement. Phenibut is hard to find at retail stores, though it’s widely available for purchase online.
After researching different products and prices, I found an awesome company online that sells high-quality phenibut for cheap. I tried it out for myself and LOVED it. Very good stuff.
I HIGHLY RECOMMEND phenibut as an effective opiate withdrawal remedy.
If you can afford it, I also highly recommend taking this awesome supplement, because the benefits are just too good to pass up.
If you have any questions on using phenibut for opiate withdrawal, please feel free to post them in the comment box below.